The Chemistry of Heterocyclic Compounds, Synthesis of Fused Heterocycles ( Chemistry of Heterocyclic Compounds: A Series Of Monographs )

Publication series :Chemistry of Heterocyclic Compounds: A Series Of Monographs

Author: Gwynn P. Ellis  

Publisher: John Wiley & Sons Inc‎

Publication year: 2009

E-ISBN: 9780470188828

P-ISBN(Hardback):  9780471914310

Subject: O626 heterocyclic compound

Language: ENG

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Description

This book classifies methods of synthesizing a heterocyclic ring which is fused to another ring. Classification is based on the functional group or groups present in the substrate, each chapter being devoted to the reactions of a particular pair of groups. The groups are arranged alphabetically so that they can be found easily. The book enables the reader to locate references (over 2000 are included) to the conversion of a wide variety of functional groups into heterocyclic rings of five to eight atoms. Each cyclization is shown as an equation which contains concise details or reagents, conditions, and yields. Since the classification of each cyclization is based on the functional groups involved, locating the relevant reference is independent of the identity of the ring in the substrate. This simplifies the search for the relevant reference.

Chapter

Contents

pp.:  1 – 9

Preface

pp.:  9 – 13

1. Introduction

pp.:  13 – 15

2. Acetal or Aldehyde and Amine

pp.:  15 – 22

4. Acylamine and Aldehyde or Ketone

pp.:  31 – 35

5. Acylamine and Amine

pp.:  35 – 38

6. Acylamine or Carbamate and Carboxamide or Nitrile

pp.:  38 – 43

7. Acylamine and Carboxylic Acid or Ester

pp.:  43 – 46

8. Acylamine or Amine and Ether or Thioether

pp.:  46 – 51

9. Acylamine, Acylhydrazine or Amine and Halogen

pp.:  51 – 54

10. Acylamine or Amine and Hydroxy or Thiol

pp.:  54 – 62

11. Acylamine, Amine or Diazonium Salt and Lactam Carbonyl

pp.:  62 – 74

12. Acylamine or Amine and Methylene

pp.:  74 – 82

13. Acylamine or Amine and Nitrile

pp.:  82 – 88

14. Acylamine, Acylhydrazine, Amine or Carbamate and Nitro

pp.:  88 – 97

15. Acylamine or Amine and Nitroso or N-oxide

pp.:  97 – 100

16. Acylamine, Acyloxy, Amine or Hydroxy and Phosphorane

pp.:  100 – 103

17. Acylamine or Acylhydrazine and Ring-carbon or Ring-sulphur

pp.:  103 – 106

18. Acylamine or Acylhydrazine and Ring-nitrogen

pp.:  106 – 112

19. Acylamine or Amine and Sulphonamide, Thioureide or Ureide

pp.:  112 – 116

20. Acylamine or Amine and Thiocyanate

pp.:  116 – 119

21. Acyl halide and Ring-carbon or Ring-nitrogen

pp.:  119 – 121

22. Aldehyde or Ketone and Alkene or Alkyne

pp.:  121 – 124

23. Aldehyde or Ketone and Azide

pp.:  124 – 127

24. Aldehyde or Ketone and Carbamate

pp.:  127 – 130

25. Aldehyde or Ketone and Carboxamide or Hydrazide

pp.:  130 – 132

26. Aldehyde or Ketone and Carboxylic Acid or Ester

pp.:  132 – 134

27. Aldehyde or Ketone and Ether or Thioether

pp.:  134 – 139

28. Aldehyde or Ketone and Halogen

pp.:  139 – 144

29. Aldehyde and Hydroxy, Thiol or Thiocyanate

pp.:  144 – 151

30. Aldehyde and Ketone; Dialdehyde or Diketone

pp.:  151 – 157

31. Aldehyde or Ketone and Methylene

pp.:  157 – 168

32. Aldehyde or Ketone and Nitrile

pp.:  168 – 171

33. Aldehyde or Ketone and Nitro, Nitroso or N-Oxide

pp.:  171 – 173

34. Aldehyde or other Carbonyl and Phosphorane

pp.:  173 – 175

35. Aldehyde or Ketone and Ring-carbon

pp.:  175 – 180

36. Aldehyde or Ketone and Ring-nitrogen

pp.:  180 – 189

37. Alkene or Alkyne and Amine or Nitro

pp.:  189 – 194

38. Alkene or Alkyne and Carboxylic Acid or its Derivative

pp.:  194 – 198

39. Alkene or Alkyne and Halogen

pp.:  198 – 201

40. Alkene or Alkyne and Hydroxy, Thiol or Ether

pp.:  201 – 203

41. Alkene, Methylene, Ring-carbon, or Ring-nitrogen and Lactam Carbonyl

pp.:  203 – 207

42. Alkene or Alkyne and Methylene, Ring-carbon or Ring-nitrogen

pp.:  207 – 211

43. Amidine and Amine, Carboxylic Acid, Ester, Hydroxy, Methylene or Nitro

pp.:  211 – 217

44. Amidine and Ring-carbon or Ring-nitrogen

pp.:  217 – 220

45. Amine and Azo or Diazo

pp.:  220 – 222

46. Amine and Carboxamide or Thiocarboxamide

pp.:  222 – 224

47. Amine and Carboxylic Acid

pp.:  224 – 233

48. Amine and Carboxylic Ester

pp.:  233 – 240

49. Amine and Enamine

pp.:  240 – 253

50. Amine and Hydrazide or Hydrazine

pp.:  253 – 255

51. Amine and Hydrazone or Imine

pp.:  255 – 260

52. Amine and Ketone

pp.:  260 – 265

53. Amine and Ring-carbon or Ring-sulphur

pp.:  265 – 276

54. Amine and Ring-nitrogen

pp.:  276 – 290

55. Azide and Azo or Nitro

pp.:  290 – 306

56. Azide and a Carboxylic Acid or its Derivative

pp.:  306 – 308

57. Azide and Methyl, Methylene or Methine

pp.:  308 – 311

58. Azide and Ring-carbon

pp.:  311 – 313

59. Azide and Ring-nitrogen

pp.:  313 – 318

60. Azo or Triazene and Carbamate, Carboxylic Acid, Ester or Nitrile

pp.:  318 – 321

61. Carbamate or Ureide and Ring-carbon or Ring-nitrogen

pp.:  321 – 323

62. Carboxamide and another Carboxylic Acid Derivative

pp.:  323 – 331

63. Carboxamide or Sulphonamide and Diazonium Salt or Diazo

pp.:  331 – 334

64. Carboxamide, Hydroxamic Acid, Hydrazide, Nitrile or Ureide and Hydroxy or Ether

pp.:  334 – 336

65. Carboxamide or Nitrile and Ring-carbon or Ring-nitrogen

pp.:  336 – 342

66. Carboxylic Acid or its Derivative and Halogen

pp.:  342 – 350

67. Carboxylic Acid or Ester and Hydrazide or Hydrazine

pp.:  350 – 361

68. Carboxylic Acid, Acyl Chloride or Ester and Hydroxy or Ether

pp.:  361 – 364

69. Carboxylic Acid or its Derivative and Lactam Carbonyl or Isocyanate

pp.:  364 – 371

70. Carboxylic Acid, Ester, Nitrile or Isonitrile and Methylene

pp.:  371 – 376

71. Carboxylic Acid Halide or Ester and Nitrile

pp.:  376 – 384

72. Carboxylic Acid, its Derivative or Lactam Carbonyl and Nitro or Ureide

pp.:  384 – 387

73. Carboxylic Acid or Ester and Ring-carbon

pp.:  387 – 392

74. Carboxylic Acid or Ester and Ring-nitrogen

pp.:  392 – 401

75. Carboxylic Acid or its Derivative and a Sulphinic or Sulphonic Acid Derivative

pp.:  401 – 408

76. 1, 2-Diamine

pp.:  408 – 412

77. 1, 3-, 1, 4-and 1, 5-Diamine

pp.:  412 – 440

78. Diazo or Diazonium Salt and Methylene

pp.:  440 – 447

79. Diazo or Diazonium Salt and Ring-carbon or Ring-nitrogen

pp.:  447 – 450

80. Dicarboxylic Acid, its Anhydride, Diacyl Halide, Diester or Dihydrazide

pp.:  450 – 456

81. Dihalogen

pp.:  456 – 460

82. Diol or Dithiol

pp.:  460 – 465

83. Dinitrile

pp.:  465 – 470

84. Di-Ring-carbon or Di-Ring-nitrogen

pp.:  470 – 472

85. Enamine and Ester or Ketone

pp.:  472 – 478

86. Enamine and a Non-carbonyl Group

pp.:  478 – 483

87. Ether or Thioether and Ring-carbon or Ring-nitrogen

pp.:  483 – 487

88. Halogen and Hydroxy or Thiol

pp.:  487 – 491

89. Halogen and Lactam Carbonyl or a Sulphur-containing Group

pp.:  491 – 499

90. Halogen and Methylene or Ring-carbon

pp.:  499 – 503

91. Halogen and Nitro

pp.:  503 – 506

92. Halogen and Ring-nitrogen

pp.:  506 – 511

93. Hydrazide or Hydrazine and Nitro or Ring-nitrogen

pp.:  511 – 517

94. Hydrazine and Ring-carbon or Ring-nitrogen

pp.:  517 – 522

95. Hydrazone or Oxime and Ring-carbon or Ring-nitrogen

pp.:  522 – 536

96. Hydroxy and Ketone or Lactam Carbonyl

pp.:  536 – 542

97. Hydroxy and Methylene

pp.:  542 – 547

98. Hydroxy and Nitro, Nitroso or Ring-nitrogen

pp.:  547 – 551

99. Hydroxy or Thiol and Ring-carbon

pp.:  551 – 554

100. Imine and Hydroxy, Ring-carbon or Ring-nitrogen

pp.:  554 – 561

101. Isocyanate or Isothiocyanate and Methylene, Ring-carbon or Ring-nitrogen

pp.:  561 – 564

102. Ketone and Lactam Carbonyl

pp.:  564 – 568

103. Methylene and Nitro or Nitroso

pp.:  568 – 572

104. Methylene and Ring-carbon or Ring-nitrogen

pp.:  572 – 576

105. Nitro or N-oxide and Ring-carbon or Ring-nitrogen

pp.:  576 – 582

106. Ring-carbon and Ring-nitrogen

pp.:  582 – 585

107. Ring-nitrogen and Thiol or Lactam Thiocarbonyl

pp.:  585 – 587

Appendix: Notes on Naming Some Fused Heterocycles

pp.:  587 – 592

List of Books and Monographs

pp.:  592 – 595

References

pp.:  595 – 597

General Index

pp.:  597 – 647

Index of Ring Systems

pp.:  647 – 653

LastPages

pp.:  653 – 675

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