Application of structure-metabolism relationships in the identification of a selective endothelin A antagonist, BMS-193884, with favourable pharmacokinetic properties

Author： Humphreys W. G.   Obermeier M. T.   Barrish J. C.   Chong S.   Marino A. M.   Murugesan N.   Wang-Iverson D.   Morrison R. A.  

Publisher： Informa Healthcare

ISSN： 1366-5928

Source： Xenobiotica, Vol.33, Iss.11, 2003-11, pp. : 1109-1123

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