Inhibitors of type 1 17β-hydroxysteroid dehydrogenase with reduced estrogenic activity: Modifications of the positions 3 and 6 of estradiol

By Tremblay Martin R.   Boivin Roch P.   Luu-The Van   Poirier Donald  

Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 20, Iss. 2, 2005-04 ,pp. : 153-163

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Chemical synthesis and in vitro biological evaluation of a phosphorylated bisubstrate inhibitor of type 3 17β-hydroxysteroid dehydrogenase

By Bérubé Marie   Poirier Donald  

Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 22, Iss. 2, 2007-04 ,pp. : 201-211

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PPARα Agonists Reduce 11β-Hydroxysteroid Dehydrogenase Type 1 in the Liver

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Improved synthesis of EM-1745, preparation of its C17-ketone analogue and comparison of their inhibitory potency on 17β-hydroxysteroid dehydrogenase type 1

By Bérubé Marie   Poirier Donald  

Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 24, Iss. 3, 2009-06 ,pp. : 832-843

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Some Coumarins and Triphenylethene Derivatives as Inhibitors of Human Testes Microsomal 17β-hydroxysteroid Dehydrogenase (17β-HSD Type 3): Further Studies with Tamoxifen on the Rat Testes Microsomal Enzyme

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Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 17, Iss. 2, 2002-01 ,pp. : 93-100

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