Evaluation of the endothelin receptor antagonists ambrisentan, darusentan, bosentan, and sitaxsentan as substrates and inhibitors of hepatobiliary transporters in sandwich-cultured human hepatocytes

Author： Hartman J. C.   Brouwer Kenneth   Mandagere Arun   Melvin Lawrence   Gorczynski Richard  

Publisher： NRC Research Press

ISSN： 1205-7541

Source： Canadian Journal of Physiology and Pharmacology, Vol.88, Iss.6, 2010-06, pp. : 682-691

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