Structural modification of an EGFR inhibitor that showed weak off-target activity against RET leading to the discovery of a potent RET inhibitor

Author： Sun Qi-Zheng   Xu Yong   Liu Jing-Jing   Zhang Chun-Hui   Wang Ze-Rong   Zheng Ren-Lin   Wang Wen-Jing   Li Lin-Li   Yang Sheng-Yong  

Publisher： Springer Publishing Company

ISSN： 1381-1991

Source： Molecular Diversity, Vol.18, Iss.2, 2014-05, pp. : 403-409

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