Publisher： John Wiley & Sons Inc
E-ISSN： 1615-4169|357|14‐15|3052-3056
ISSN： 1615-4150
Source： ADVANCED SYNTHESIS & CATALYSIS, Vol.357, Iss.14‐15, 2015-10, pp. : 3052-3056
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Abstract
AbstractAn efficient catalytic approach to the synthesis of N,N‐dialkyl‐2‐alkynylanilines was developed by using Pd‐catalyzed norbornene‐mediated three‐component reactions of haloarenes, alkoxyamines (RO‐NR2), and alkynes. The procedure forms one CN bond and one CC bond efficiently in a one‐pot manner from readily available starting materials. A number of 2‐alkynylanilines with a broad range of functional groups were afforded in good to excellent yields.
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