Site-directed mutagenesis of the 5-HT 1B receptor increases the affinity of 5-HT for the agonist low-affinity conformation and reduces the intrinsic activity of 5-HT

By Granas C.   Nordquist J.   Mohell N.   Larhammar D.  

European Journal of Pharmacology, Vol. 421, Iss. 2, 2001-06 ,pp. : 69-76

Elsevier

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Site-directed mutagenesis of the putative human muscarinic M 2 receptor binding site

By Heitz F.   Holzwarth J.A.   Gies J.-P.   Pruss R.M.   Trumpp-Kallmeyer S.   Hibert M.F.   Guenet C.  

European Journal of Pharmacology, Vol. 380, Iss. 2, 1999-09 ,pp. : 183-195

Elsevier

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Site-directed mutagenesis of the human adenosine A 2A receptor. Critical involvement of Glu 13 in agonist recognition

By IJzerman A.P.   Kunzel J.K.V.F.D.   Kim J.   Qiaoling J.   Jacobson K.A.  

European Journal of Pharmacology, Vol. 310, Iss. 2, 1996-08 ,pp. : 269-272

Elsevier

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SB-236057, a selective 5-HT 1B receptor inverse agonist, blocks the 5-HT human terminal autoreceptor

By Middlemiss D.N.   Gothert M.   Schlicker E.   Scott C.M.   Selkirk J.V.   Watson J.   Gaster L.M.   Wyman P.   Riley G.   Price G.W.  

European Journal of Pharmacology, Vol. 375, Iss. 1, 1999-06 ,pp. : 359-365

Elsevier

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5-HT 1B/D Receptor Antagonists

By Pauwels P.J.  

General Pharmacology, Vol. 29, Iss. 3, 1997-09 ,pp. : 293-303

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