Assessing and minimizing time-dependent inhibition of cytochrome P450 3A in drug discovery: A case study with melanocortin-4 receptor agonists

Author： Tang W.   Stearns R. A.   Wang R. W.   Miller R. R.   Chen Q.   Ngui J.   Bakshi R. K.   Nargund R. P.   Dean D. C.   Baillie T. A.  

Publisher： Informa Healthcare

ISSN： 1366-5928

Source： Xenobiotica, Vol.38, Iss.11, 2008-11, pp. : 1437-1451

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