A fission yeast-based test system for the determination of IC₅₀ values of anti-prostate tumor drugs acting on CYP21

By Drăgan Călin-Aurel   Hartmann Rolf W.   Bureik Matthias  

Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 21, Iss. 5, 2006-10 ,pp. : 547-556

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IC₅₀-based approaches as an alternative method for assessment of time-dependent inhibition of CYP3A4

By Burt Howard J.   Galetin Aleksandra   Houston J. Brian  

Xenobiotica, Vol. 40, Iss. 5, 2010-05 ,pp. : 331-343

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Validation of cytochrome P450 time-dependent inhibition assays: a two-time point IC50 shift approach facilitates kinact assay design

By Perloff E. S.   Mason A. K.   Dehal S. S.   Blanchard A. P.   Morgan L.   Ho T.   Dandeneau A.   Crocker R. M.   Chandler C. M.   Boily N.   Crespi C. L.   Stresser D. M.  

Xenobiotica, Vol. 39, Iss. 2, 2009-02 ,pp. : 99-112

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Synthesis, characterization and inhibitory potency of two oxono and thiono analogues of phosphoramidate compounds on acetylcholinesterase

By Gholivand Khodayar   Mojahed Fresia   Salehi Marjan   Naderi-Manesh Hossein   Khajeh Khosro  

Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 21, Iss. 5, 2006-10 ,pp. : 521-525

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Synthesis of a novel series of bispyridinium compounds bearing a xylene linker and evaluation of their reactivation activity against chlorpyrifos-inhibited acetylcholinesterase

By Musilek K.   Kuca K.   Jun D.   Dohnal V.   Dolezal M.  

Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 20, Iss. 5, 2005-10 ,pp. : 409-415

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