Synthesis and Biological Evaluation of Estradiol-Core Derivatives Bearing a Fused &ggr;-Lactone as Inhibitors of 17&bgr;-Hydroxysteroid Dehydrogenase Type 1

Publisher： Bentham Science Publishers

E-ISSN： 1875-6662|10|1|39-53

ISSN： 1573-4080

Source： Current Enzyme Inhibition, Vol.10, Iss.1, 2014-05, pp. : 39-53

Disclaimer: Any content in publications that violate the sovereignty, the constitution or regulations of the PRC is not accepted or approved by CNPIEC.

Previous Menu Next

Abstract

Related content

Structure and Inhibitor Binding Mechanisms of 11&bgr; -Hydroxysteroid Dehydrogenase Type 1

By  

Current Chemical Biology, Vol. 3, Iss. 2, 2009-05 ,pp. : 159-170

Bentham Science Publishers

Access to resources Recommend Favorite

Inhibitors of type 1 17β-hydroxysteroid dehydrogenase with reduced estrogenic activity: Modifications of the positions 3 and 6 of estradiol

By Tremblay Martin R.   Boivin Roch P.   Luu-The Van   Poirier Donald  

Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 20, Iss. 2, 2005-04 ,pp. : 153-163

Informa Healthcare

Access to resources Recommend Favorite

Chemical synthesis and in vitro biological evaluation of a phosphorylated bisubstrate inhibitor of type 3 17β-hydroxysteroid dehydrogenase

By Bérubé Marie   Poirier Donald  

Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 22, Iss. 2, 2007-04 ,pp. : 201-211

Informa Healthcare

Access to resources Recommend Favorite

Synthesis and Evaluation of Amido-Deoxyestradiol Derivatives as Inhibitors of 17&bgr;-Hydroxysteroid Dehydrogenase Type 12

By  

Current Enzyme Inhibition, Vol. 7, Iss. 3, 2011-10 ,pp. : 134-146

Bentham Science Publishers

Access to resources Recommend Favorite

Direct antiproliferative effect of nonsteroidal 17β-hydroxysteroid dehydrogenase type 1 inhibitors in vitro

By Berényi Ágnes  

Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 28, Iss. 4, 2013-08 ,pp. : 695-703

Informa Healthcare

Access to resources Recommend Favorite